https://vital.seals.ac.za/vital/access/manager/Index ${session.getAttribute("locale")} 5 Synthesis and anti-parasitic activity of C-benzylated (N-arylcarbamoyl) alkylphosphonate esters https://vital.seals.ac.za/vital/access/manager/Repository/vital:35803 Wed 12 May 2021 22:21:55 SAST ]]> Identification of Novel Potential Inhibitors of Pteridine Reductase 1 in Trypanosoma brucei via Computational Structure-Based Approaches and in Vitro Inhibition Assays https://vital.seals.ac.za/vital/access/manager/Repository/vital:35647 Wed 12 May 2021 19:28:13 SAST ]]> In vitro antimalarial, antitrypanosomal and HIV-1 integrase inhibitory activities of two Cameroonian medicinal plants: Antrocaryon klaineanum (Anacardiaceae) and Diospyros conocarpa (Ebenaceae) https://vital.seals.ac.za/vital/access/manager/Repository/vital:35908 Wed 12 May 2021 18:58:35 SAST ]]> Synthesis and evaluation of substituted 4-(N-benzylamino)cinnamate esters as potential anti-cancer agents and HIV-1 integrase inhibitors https://vital.seals.ac.za/vital/access/manager/Repository/vital:28929 Wed 12 May 2021 18:24:55 SAST ]]> Cinnamoyl-Oxaborole Amides: Synthesis and Their in Vitro Biological Activity. https://vital.seals.ac.za/vital/access/manager/Repository/vital:35362 125 μM) was observed. Similarly, these compounds exhibited moderate activity against the human protozoal pathogen Trichomonas vaginalis with no observed effect on common microbiome bacterial species. The cross-species inhibitory activity presents the possibility of these compounds serving as broad-spectrum antibiotics for these prevalent three human pathogens.]]> Wed 12 May 2021 17:39:06 SAST ]]> In vitro Anti-trypanosomal activities of indanone-based chalcones: https://vital.seals.ac.za/vital/access/manager/Repository/vital:40169 Wed 12 May 2021 14:54:55 SAST ]]> Synthesis, structure and in vitro anti-trypanosomal activity of non-toxic Arylpyrrole-Based Chalcone derivatives: https://vital.seals.ac.za/vital/access/manager/Repository/vital:40096 Wed 12 May 2021 14:50:45 SAST ]]> Detection of the in vitro modulation of Plasmodium falciparum Arf1 by Sec7 and ArfGAP domains using a colorimetric plate-based assay: https://vital.seals.ac.za/vital/access/manager/Repository/vital:41242 Wed 12 May 2021 14:45:45 SAST ]]> NMR structural elucidation of channaine, an unusual alkaloid from Sceletium tortuosum: https://vital.seals.ac.za/vital/access/manager/Repository/vital:41110 Wed 12 May 2021 14:36:55 SAST ]]> A New Synthetic Method for Tetraazatricyclic Derivatives and Evaluation of Their Biological Properties https://vital.seals.ac.za/vital/access/manager/Repository/vital:35413 Wed 05 Apr 2023 08:51:09 SAST ]]> Synthesis, characterization and biological activity of some Dithiourea Derivatives: https://vital.seals.ac.za/vital/access/manager/Repository/vital:41007 Wed 05 Apr 2023 08:50:35 SAST ]]> Biological activity of plant extracts and isolated compounds from Alchornea laxiflora: Anti-HIV, antibacterial and cytotoxicity evaluation https://vital.seals.ac.za/vital/access/manager/Repository/vital:35907 Wed 04 Aug 2021 14:30:34 SAST ]]> Anti-HIV-1 integrase potency of methylgallate from Alchornea cordifolia using in vitro and in silico approaches: https://vital.seals.ac.za/vital/access/manager/Repository/vital:41001 Wed 04 Aug 2021 14:30:33 SAST ]]> Application of the Morita-Baylis-Hillman reaction in the synthesis of 3-[(N-cycloalkylbenzamido)methyl]-2-quinolones as potential HIV-1 integrase inhibitors https://vital.seals.ac.za/vital/access/manager/Repository/vital:28913 Tue 31 Aug 2021 12:27:45 SAST ]]> Synthesis, in vitro cytotoxicity and trypanocidal evaluation of novel 1, 3, 6-substituted non-fluoroquinolones https://vital.seals.ac.za/vital/access/manager/Repository/vital:35409 Tue 31 Aug 2021 12:26:10 SAST ]]> Synthesis, antiplasmodial and antitrypanosomal evaluation of a series of novel 2-oxoquinoline-based thiosemicarbazone derivatives https://vital.seals.ac.za/vital/access/manager/Repository/vital:35407 50 % was often observed. Except for compound 9o, none of the final compounds exhibited cytotoxic effects against HeLa cells at 20 μM.]]> Tue 31 Aug 2021 12:24:51 SAST ]]> New thiazolidine-2,4-dione derivatives combined with organometallic ferrocene: Synthesis, structure and antiparasitic activity https://vital.seals.ac.za/vital/access/manager/Repository/vital:35382 90% viability of the HeLa cell line screened.]]> Tue 31 Aug 2021 12:24:00 SAST ]]> Quinolone-isoniazid hybrids: Synthesis and preliminary in vitro cytotoxicity and anti-tuberculosis evaluation https://vital.seals.ac.za/vital/access/manager/Repository/vital:35410 Tue 31 Aug 2021 12:20:16 SAST ]]> Terminaliamide, a new ceramide and other phytoconstituents from the roots of Terminalia mantaly H. Perrier and their biological activities https://vital.seals.ac.za/vital/access/manager/Repository/vital:45422 Tue 30 Nov 2021 15:50:54 SAST ]]> Compounds isolation and biological activities of Piptadeniastrum africanum (hook. f.) Brennan (Fabaceae) roots: https://vital.seals.ac.za/vital/access/manager/Repository/vital:38938 Tue 09 Aug 2022 06:12:33 SAST ]]> Potential repurposing of four FDA approved compounds with antiplasmodial activity identified through proteome scale computational drug discovery and in vitro assay https://vital.seals.ac.za/vital/access/manager/Repository/vital:42830 Tue 09 Aug 2022 05:58:00 SAST ]]> The in vitro antiplasmodial and antiproliferative activity of new ferrocene-based α-aminocresols targeting hemozoin inhibition and DNA interaction: https://vital.seals.ac.za/vital/access/manager/Repository/vital:38827 Thu 26 Aug 2021 14:51:36 SAST ]]> Repurposing a polymer precursor: Synthesis and in vitro medicinal potential of ferrocenyl 1, 3-benzoxazine derivatives https://vital.seals.ac.za/vital/access/manager/Repository/vital:41240 Thu 26 Aug 2021 14:44:36 SAST ]]> Biological activities of plant extracts from Ficus elastica and Selaginella vogelli: an antimalarial, antitrypanosomal and cytotoxity evaluation https://vital.seals.ac.za/vital/access/manager/Repository/vital:35853 Thu 13 May 2021 06:37:22 SAST ]]> Indolyl-3-ethanone-α-thioethers: a promising new class of non-toxic antimalarial agents https://vital.seals.ac.za/vital/access/manager/Repository/vital:28920 Thu 13 May 2021 04:21:40 SAST ]]> Plasmodium falciparum Hep1 is required to prevent the self aggregation of PfHsp70-3 https://vital.seals.ac.za/vital/access/manager/Repository/vital:28903 Thu 11 Aug 2022 06:48:12 SAST ]]> Ferrocenyl and organic novobiocin derivatives: synthesis and their in vitro biological activity https://vital.seals.ac.za/vital/access/manager/Repository/vital:28914 Thu 07 Jul 2022 21:23:26 SAST ]]> Expanding the SAR of Nontoxic Antiplasmodial Indolyl-3-ethanone Ethers and Thioethers: https://vital.seals.ac.za/vital/access/manager/Repository/vital:41114 Thu 07 Jul 2022 21:23:25 SAST ]]> Novobiocin–ferrocene conjugates possessing anticancer and antiplasmodial activity independent of HSP90 inhibition. https://vital.seals.ac.za/vital/access/manager/Repository/vital:35359 Thu 07 Jul 2022 21:23:25 SAST ]]> Dynamic mitochondrial localisation of STAT3 in the cellular adipogenesis model 3T3-L1: https://vital.seals.ac.za/vital/access/manager/Repository/vital:41181 Mon 13 Nov 2023 20:30:05 SAST ]]> Expanding the SAR of Nontoxic Antiplasmodial Indolyl-3-ethanone Ethers and Thioethers. https://vital.seals.ac.za/vital/access/manager/Repository/vital:35370 Fri 03 Dec 2021 18:29:07 SAST ]]>